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Effects of FK506 on Ca(2+) Release Channels (Review)

Tacrolimus (FK506), which was isolated from the fermentation broth of Streptomyces tsukubaensis No. 9993, has an immunosuppressive effect. In T-lymphocytes, FK506 binds to the intracellular receptor, a 12-kDa FK506-binding protein (FKBP12). The FK506-FKBP12 complex binds to the phosphatase calcineur...

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Autor principal: Ozawa, Terutaka
Format: Article
Idioma:English
Publicat: Libertas Academica 2008
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC2746578/
https://ncbi.nlm.nih.gov/pubmed/19787097
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