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Potent, structurally constrained agonists and competitive antagonists of corticotropin-releasing factor.

Predictive methods, physicochemical measurements, and structure activity relationship studies suggest that corticotropin-releasing factor (CRF; corticoliberin), its family members, and competitive antagonists (resulting from N-terminal deletions) usually assume an alpha-helical conformation when int...

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Main Authors: Gulyas, J, Rivier, C, Perrin, M, Koerber, S C, Sutton, S, Corrigan, A, Lahrichi, S L, Craig, A G, Vale, W, Rivier, J
格式: Artigo
語言:en
出版: 1995
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在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC40654/
https://ncbi.nlm.nih.gov/pubmed/7479843
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