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Inhibition of Antibiotic Efflux in Bacteria by the Novel Multidrug Resistance Inhibitors Biricodar (VX-710) and Timcodar (VX-853)

Inhibitors of mammalian multidrug efflux, such as the plant alkaloid reserpine, are also active in potentiating antibiotic activity by inhibiting bacterial efflux. Based on this precedent, two novel mammalian multiple drug resistance inhibitors, biricodar (VX-710) and timcodar (VX-853), were evaluat...

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Autores principales: Mullin, Steve, Mani, Nagraj, Grossman, Trudy H.
Formato: Artículo
Lenguaje:English
Publicado: American Society for Microbiology 2004
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC525397/
https://ncbi.nlm.nih.gov/pubmed/15504837
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.48.11.4171-4176.2004
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