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Second-generation inhibitors of Bruton tyrosine kinase
Abstract Bruton tyrosine kinase (BTK) is a critical effector molecule for B cell development and plays a major role in lymphoma genesis. Ibrutinib is the first-generation BTK inhibitor. Ibrutinib has off-target effects on EGFR, ITK, and Tec family kinases, which explains the untoward effects of ibru...
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| Publicado en: | Journal of Hematology & Oncology |
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| Autores principales: | , , , |
| Formato: | Artículo |
| Publicado: |
BMC
2016-09-01
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| Acceso en línea: | http://link.springer.com/article/10.1186/s13045-016-0313-y |
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